The Ultimate Guide to Toremifene Citrate

Chances are you’re zeroing in for ways to make the most out of your post cycle therapy if you are logging on to the worldwide web and looking up Toremifene Citrate. Also known in the bodybuilding world as Torem and Fareston, it’s not just by sheer coincidence why it has become one of the most popular post cycle therapy or PCT go-to drugs these days, too.

Are you ready to take your Toremifene Citrate know-how up a notch? Make sure you follow along to get the lowdown on all the important details you need to know about it so you can easily make an informed decision if this one should be in your arsenal after your cycle.

So What Exactly is Toremifene Citrate?

Toremifene Citrate is essentially a non-steroidal anti-estrogen drug that is derived from triphenylethylene, which is a type of hydrocarbon that has been discovered to possess estrogenic effects in 1937.

Now while Torem has made a name for itself in bodybuilding circles over the years as a PCT drug, it was originally developed to help treat breast cancer in postmenopausal women, particularly in cases where the disease is on the verge of spreading or has already spread to other parts of the body.

Toremifene Citrate chemical structure

The brand name Fareston was first patented by the Finnish company, Orion Corporation, and got the green light to be marketed as a cancer treatment sometime in the mid 1990’s. It made its way to the United States via the distribution and marketing of Roberts Pharma just a few years later.

Moreover, Torem is also capable of cutting off the effects of estrogen in and around the breast tissue that can be vulnerable to cancer by fooling its receptors. This is the upshot that has propelled this drug to become an essential when PCT is concerned. There are also scientific studies that show Torem is less toxic compared to Nolvadex when used for post cycle therapy.

Belonging to a class of drugs known as selective estrogen receptor modulators or SERM’s, Toremifene Citrate basically binds to the receptors of estrogen to trigger a boost in androgens or male hormones, particularly testosterone, after running an anabolic cycle. We will touch more on this shortly.

How does Toremifene Citrate Work?

After running an anabolic cycle, the amounts of follicle-stimulating hormones (FSH) and luteinizing hormones (LH) produced in your body plummet until they reach critical levels. It is even possible that their production rates are completely shut down during the same, which leads to a deficit in testosterone and a surplus in estrogen.

Although a surge in estrogen hormones is considered normal after a cycle, the side effects that you can go through if this issue isn’t set right as soon as possible can be rather detrimental not just for the gains that you’ve been able to realize, but also to your overall health.

Besides putting you at risk for erratic blood pressure levels, lethargic episodes and unwanted water retention, you can be also in for “bitch tits” or gynecomastia, which I’m pretty sure isn’t one of the things that you’ve got in mind when you started running a cycle in the first place. This is the biggest reason why a proper post cycle therapy should be in your checklist.

Example of gynecomastia or “bitch tits,” a side effect of having excessive estrogen levels.

Moving on, Toremifene Citrate helps jumpstart normal testosterone production in the body by binding to the receptors of estrogen hormones to prevent them from making their way to the pituitary gland. This makes the body think that estrogen levels are up to par and stimulates the hypothalamic-pituitary-testicular axis or the HPTA, for short, to kick in and start producing testosterone again.

Toremifene Citrate Half-Life

The term “half-life” simply means the duration when it gets eliminated from the bloodstream. Scientific studies show that the half-life of Toremifene Citrate is approximately 5 days, which is similar to other PCT drugs like Nolvadex and Clomid.

Toremifene Citrate Dosing Suggestions

Knowing your ideal Toremifene Citrate dosing plays a very important role in terms of achieving the results you want, whether you’re planning to use it as an on-cycle drug or perhaps for post cycle therapy. We’ve come up with a quick walkthrough below to make things easier for you.

On-cycle usage:

Experts recommend a dose of 30 to 60 milligrams daily if you’re using Torem as an on-cycle drug for the prevention of gynecomastia or “bitch tits.” But the thing is it’s really important to take note that if gynecomastia is already developing or has already developed during the same, a dose of 120 milligrams should be taken along with an aromatase inhibitor.

PCT usage:

According to seasoned anabolic steroid users, a daily dose of 120 milligrams of Toremifene Citrate should be taken for the first week of post cycle therapy. For the second week, it should be tapered down to 100 milligrams. For the remaining third and fourth week of PCT, 60 milligrams of Torem should be administered.

Interestingly, there are no special considerations to keep an eye on when using Toremifene Citrate. You can take it before, during, or following meals and can be administered either during the morning or evening. There is no need to split the doses throughout the day as well.

Toremifene Citrate Side Effects

Akin to other pharmaceutical products, Torem has its share of side effects, albeit scientific studies show that the possibility of them occurring is lower compared to its counterparts. Some of the side effects that could be experienced during the administration of Toremifene Citrate include dizzy spells, rashes, dry eyes, bouts of vomiting and nausea, sweating, mood swings, and swelling of the extremities.

However, experts explain that it is possible that Torem can spike sex hormone binding globulin or SHBG levels during administration. When the amount of SHBG in the male body rises, the system reacts by lowering the amount of free testosterone, which can affect the total levels of testosterone produced. This can potentially lead to negative issues in terms of recovery, gains achieved and strength levels.

On the other hand, scientific studies also show that Toremifene Citrate doesn’t affect Insulin-like Growth Factor 1 or IGF-1 levels. Also called as Somatomedin C, IGF-1 plays a key role in joint health and muscle building. Its counterpart, Nolvadex, has been seen to bring down IGF-1 levels when administered.

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