The Ultimate Guide to Exemestane

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When it comes to achieving the physique that you’ve always wanted, Exemestane – or Aromasin as it is more popularly known in the bodybuilding world – is definitely one of the most crucial things to have in your checklist.

Sure you may already have a lineup of the best gear and stacks available these days at your disposal, but the thing is you’re just in for a surprise (and not the good kind either) the least you expect it when you leave out Exemestane in the whole picture.

If you’re still having second thoughts about adding Exemestane in your lineup or perhaps looking to boost your know-how about this drug, then you’ve come to the right place. Make sure you follow along to find out why cycling without this bodybuilding essential is no doubt one of the biggest mistakes that you’ll ever make.

Getting to Know Exemestane

At its simplest, Exemestane is a type of drug that helps control an unwanted enzyme called aromatase that usually makes an appearance in the tissues of the male body when cycling with steroids. It is usually used as an on-cycle estrogen control drug and during post-cycle therapy (PCT).

Aromatase basically converts the muscle-building testosterone to the female hormone estrogen. A surplus of estrogen in the body can lead to nasty side effects like excessive water retention, surges in blood pressure levels, lethargy, as well as gynecomastia or the undesirable growth of male breast tissue, if not properly suppressed.

Exemestane belongs to the aromatase inhibitor or AI class of drugs, which also includes Arimidex and Letrozole. However, what makes Exemestane really special when compared to its counterparts is the fact that it is a “suicidal” AI. This simply means that it will disable the aromatase enzyme for good as soon as it binds to it.

Although Arimidex and Letrozole also have the ability to suppress aromatase by themselves, they only work as long as you’re taking them. When you stop using these AI’s, this eventually triggers a negative effect called “estrogen rebound” that makes you prone yet again to the nasty issues that take place when the estrogen levels in your body spike.

A Brief History on Exemestane

While Exemestane has already established its mettle over the years as a key component of an ideal anabolic cycle, especially when steroids are involved, it was originally formulated to help prevent and treat breast cancer among post-menopausal women.

The chemical structure of Exemestane

Pharmacia & Upjohn is deemed as the original manufacturer of Exemestane, but Pfizer is the main distributor of the same ever since it was given the green light by the FDA in 1999.

Exemestane Half-Life

According to experts, Exemestane has a fairly short half-life of 9 hours in men – compared to 27 hours in women – and dissipates rather quickly as soon as it is ingested. But don’t let this AI’s speedy release from the body fool you. Scientific studies show that Exemestane is capable of eliminating up to 90% of aromatase enzymes after administration.

Moreover, what’s really interesting is Exemestane is still very much potent up to 72 hours after taking a single 25mg dose. It is proven to keep baseline estrogen levels below 40% after 3 days post administration. And that’s during the time when it is almost eliminated from the body!

It is important to take note, though, that baseline estrogen levels usually returned to normal after 120 hours after administration of Exemestane, but without the risk of rebounding in any way compared to other aromatase inhibitors that you can get your hands on these days.

Exemestane Dosage

The ideal Exemestane dosage can vary from one person to another and greatly depends on the anabolic compounds that are cycled.

In the case of running a cycle with dry compounds, such as Winstrol and Masteron, the recommended dosage is around 12.5mg daily or every other day. However, if you’re cycling with wet compounds like Deca Durabolin and Dianabol, a higher dosage of 25mg is recommended.

However, if you’re really looking to gauge the most ideal Exemestane dosage that you should use during your cycle or for PCT, the best way to go is having blood work done.

Exemestane Notes

To make things even more interesting, besides being seen to boost overall testosterone levels by as much as 60% in just 10 days, Exemestane is also proven to perk up the amount of usable or free testosterone in the body while at it. How’s that for a finale?

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